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Eplerenone
Eplerenone

2.55
Action involves inhibiting aldosterone receptors to support fluid regulation and cardiac function.
Ingredient
Eplerenone
Category
Heart & Blood Pressure
Availability
In Stock
Delivery Time
Airmail (14-21 days) | Trackable (5-9 days)
Shipped in a discreet, unmarked envelope with all required documents enclosed.

Product Sheet

Active Ingredient(s)
Eplerenone
Reference Brand
Inspra
Product Origin
Generic Product
Reference Manufacturer
Pfizer
Product Form
Tablet
Regulatory Classification
Rx
Primary Category
Heart & Blood Pressure
Product Category
Aldosterone Receptor Antagonist
Pharmacological Class
Potassium-Sparing Diuretic
Manufacturer Description
Intended for heart failure to manage fluid balance and support cardiac survival post-infarction.
Mechanism of Action
Eplerenone selectively inhibits the mineralocorticoid receptor. This blocks the binding of aldosterone, which prevents sodium reabsorption and potassium excretion, effectively reducing blood pressure and myocardial fibrosis.
Route of Administration
Oral
Onset Time
1–2 weeks
Duration
4–6 hours (half-life)
Contraindications
Hyperkalemia, Severe renal impairment, Concurrent use of strong CYP3A4 inhibitors
Severe Adverse Events
Severe hyperkalemia, Renal failure, Angioedema — requires immediate medical attention
Common Side Effects
Dizziness, Fatigue, Headache
Uncommon Side Effects
Hyperkalemia, Diarrhea, Abdominal pain
Drug Interactions
Alcohol, Lithium, Potassium Supplements, Ketoconazole, ACE Inhibitors
Pregnancy Safety Warnings
FDA Category B: No evidence of fetal risk. Breastfeeding: Not known if excreted in milk.
Age Restrictions
Safety and efficacy in pediatric patients have not been established.
Storage Guidelines
Store at room temperature.
Related Products
Inspra, Aldactone, Eptus
Information related to Eplerenone is compiled and periodically reviewed with reference to established medical sources and prescribing guidance. Content is provided for general reference and should be confirmed with a registered healthcare professional before use.
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