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Ketoconazole
Ketoconazole

0.78
Helps with the disruption of fungal cell membrane integrity.
Ingredient
Ketoconazole
Category
Antifungals
Availability
In Stock
Delivery Time
Airmail (14-21 days) | Trackable (5-9 days)
Shipped in a discreet, unmarked envelope with all required documents enclosed.

Product Sheet

Active Ingredient(s)
Ketoconazole
Reference Brand
Nizoral
Product Origin
Generic Product
Reference Manufacturer
Janssen Pharmaceuticals
Product Form
Tablet, Cream, Shampoo
Regulatory Classification
Rx
Primary Category
Antifungals
Product Category
Imidazole Antifungal
Pharmacological Class
Azole Antifungal
Manufacturer Description
Utilized for systemic fungal infections to manage fungal survival and support infection clearance.
Mechanism of Action
Ketoconazole inhibits the synthesis of ergosterol by blocking the enzyme 14-alpha-demethylase. This disrupts the fungal cell membrane structure and function, eventually leading to cell death.
Route of Administration
Oral
Onset Time
1–2 days
Duration
8 hours (half-life)
Contraindications
Acute or chronic liver disease, Hypersensitivity to ketoconazole, Concurrent use of simvastatin
Severe Adverse Events
Hepatotoxicity, Qt prolongation, Adrenal insufficiency — requires immediate medical attention
Common Side Effects
Nausea, Headache, Abdominal pain
Uncommon Side Effects
Gynecomastia, Impotence, Dizziness
Drug Interactions
Alcohol, Warfarin, Rifampin, Antacids, Digoxin
Pregnancy Safety Warnings
FDA Category C: Benefit must justify risk. Breastfeeding: Excreted in milk; monitor infant.
Age Restrictions
Safety and efficacy established in pediatric patients two years and older.
Storage Guidelines
Store at room temperature and protect from light.
Related Products
Nizoral, Sporanox, Diflucan
Information related to Ketoconazole is compiled and periodically reviewed with reference to established medical sources and prescribing guidance. Content is provided for general reference and should be confirmed with a registered healthcare professional before use.
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