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Orap
Orap

0.71
Helps with the regulation of neurological impulses for neurological stability.
Ingredient
Pimozide
Category
Mental Health
Availability
In Stock
Delivery Time
Airmail (14-21 days) | Trackable (5-9 days)
Shipped in a discreet, unmarked envelope with all required documents enclosed.

Product Sheet

Active Ingredient(s)
Pimozide
Reference Brand
Pimozide
Product Origin
Generic Alternative
Reference Manufacturer
Teva Pharmaceutical Industries
Product Form
Tablet
Regulatory Classification
Rx
Primary Category
Mental Health
Product Category
First-Generation Antipsychotic
Pharmacological Class
Diphenylbutylpiperidine
Clinical Indications
Tourette syndrome, Schizophrenia
Manufacturer Description
Utilized for tourette syndrome to manage motor and vocal tics and support behavioral stability.
Mechanism of Action
Pimozide acts as a selective antagonist at dopamine D2 receptors in the central nervous system. This blocks dopamine-mediated neurotransmission in the basal ganglia, effectively reducing the frequency and severity of tics.
Route of Administration
Oral
Onset Time
1–2 weeks
Duration
55 hours (half-life)
Contraindications
Congenital long QT syndrome, History of cardiac arrhythmias, Concurrent use of CYP3A4 inhibitors, Severe CNS depression
Severe Adverse Events
Qt prolongation, Neuroleptic malignant syndrome, Tardive dyskinesia — requires immediate medical attention
Common Side Effects
Somnolence, Dry mouth, Constipation
Uncommon Side Effects
Extrapyramidal symptoms, Akathisia, Headache
Drug Interactions
Alcohol, Amiodarone, Ketoconazole, Clarithromycin, Fluoxetine
Pregnancy Safety Warnings
FDA Category C: Use only if clearly needed. Breastfeeding: Not recommended.
Age Restrictions
Safety and efficacy established in pediatric patients 12 years and older.
Storage Guidelines
Store at room temperature.
Related Products
Haldol, Largactil, Risperdal
Information related to Orap is compiled and periodically reviewed with reference to established medical sources and prescribing guidance. Content is provided for general reference and should be confirmed with a registered healthcare professional before use.
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