Sumatriptan
Sumatriptan

2.91
Reduces cranial nerve sensitivity associated with intense pressure and sensory discomfort.


Ingredient
Category
Availability
In Stock
Delivery Time
Airmail (14-21 days) | Trackable (5-9 days)
Shipped in a discreet, unmarked envelope with all required documents enclosed.

Product Sheet

Active Ingredient(s)
Sumatriptan
Reference Brand
Imitrex
Product Origin
Generic Product
Reference Manufacturer
GlaxoSmithKline
Product Form
Tablet, Nasal Spray, Injectable Solution
Regulatory Classification
Rx
Primary Category
Neurology
Product Category
Serotonin 5-HT1 Receptor Agonist
Pharmacological Class
Triptan
Clinical Indications
Manufacturer Description
Formulated for migraine and cluster headaches to alleviate acute pain and manage cranial discomfort.
Mechanism of Action
Sumatriptan binds selectively to 5-HT1B and 5-HT1D receptors on intracranial blood vessels and sensory nerves. This action results in vasoconstriction and inhibition of pro-inflammatory neuropeptide release.
Route of Administration
Oral
Onset Time
30–60 minutes
Duration
2–4 hours
Contraindications
Ischemic heart disease, Coronary vasospasm, Uncontrolled hypertension, Concurrent use of MAO inhibitors
Severe Adverse Events
Myocardial infarction, Serotonin syndrome, Stroke — requires immediate medical attention
Common Side Effects
Tingling, Flushing, Dizziness
Uncommon Side Effects
Chest tightness, Nausea, Feeling of heaviness
Drug Interactions
Alcohol, MAO Inhibitors, Ergotamine, SSRI Antidepressants, Lithium
Pregnancy Safety Warnings
FDA Category C: Use with caution. Breastfeeding: Excreted in milk; wait 12 hours after dose to nurse.
Age Restrictions
Safety and efficacy in pediatric patients under 18 years have not been established for oral use.
Storage Guidelines
Store at room temperature away from light.
Related Products
Imigran, Zomig, Relpax
Information related to Sumatriptan is compiled and periodically reviewed with reference to established medical sources and prescribing guidance. Content is provided for general reference and should be confirmed with a registered healthcare professional before use.
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