Zolmitriptan
Zolmitriptan

55.08
Regular use helps relieve migraine pain and pressure.


Ingredient
Category
Availability
In Stock
Delivery Time
Airmail (14-21 days) | Trackable (5-9 days)
Shipped in a discreet, unmarked envelope with all required documents enclosed.

Product Sheet

Active Ingredient(s)
Zolmitriptan
Reference Brand
Zomig
Product Origin
Generic Product
Reference Manufacturer
AstraZeneca
Product Form
Tablet, Orally Disintegrating Tablet, Nasal Spray
Regulatory Classification
Rx
Primary Category
Neurology
Product Category
Serotonin 5-HT1 Receptor Agonist
Pharmacological Class
Triptan
Clinical Indications
Manufacturer Description
Utilized for migraine headaches to alleviate acute symptoms and manage cranial discomfort.
Mechanism of Action
Zolmitriptan binds with high affinity to 5-HT1B and 5-HT1D receptors. This leads to the constriction of dilated cranial blood vessels and inhibits the release of pro-inflammatory neuropeptides from the trigeminal nerve.
Route of Administration
Oral
Onset Time
45–60 minutes
Duration
3 hours (half-life)
Contraindications
Ischemic heart disease, Uncontrolled hypertension, History of stroke, Concurrent use of MAO inhibitors
Severe Adverse Events
Myocardial infarction, Serotonin syndrome, Stroke — requires immediate medical attention
Common Side Effects
Tingling, Dizziness, Fatigue
Uncommon Side Effects
Chest tightness, Nausea, Dry mouth
Drug Interactions
Alcohol, MAO Inhibitors, Cimetidine, Fluoxetine, Ergotamine
Pregnancy Safety Warnings
FDA Category C: Benefit must justify risk. Breastfeeding: Excretion in milk is unknown; compatible with caution.
Age Restrictions
Safety and efficacy in pediatric patients have not been established for oral use.
Storage Guidelines
Store at room temperature away from moisture.
Related Products
Zomig, Imigran, Relpax
Information related to Zolmitriptan is compiled and periodically reviewed with reference to established medical sources and prescribing guidance. Content is provided for general reference and should be confirmed with a registered healthcare professional before use.
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